Pentamidine isethionate salt, powder

Code: P0547-25MG D2-231

Application

Antimicrobial against Pneumocystis carinii.

Pentamidine isethionate salt has been used:as a positive control for anti-leishmanial, anti-plasmodial ...


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€51.35 25MG
€63.16 inc. VAT
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Application

Antimicrobial against Pneumocystis carinii.

Pentamidine isethionate salt has been used:as a positive control for anti-leishmanial, anti-plasmodial and cytotoxic assaysas a prototypical compound to analyse the inhibitor effect on human ether-a-go-go-related gene (HERG) K+ channel traffickingas an anti-leishmanial agent in promastigotes

Biochem/physiol Actions

Pentamidine isethionate is used as a second line drug for leishmaniasis.

Neuroprotective; inhibits constitutive nitric oxide synthase in the brain; NMDA glutamate receptor antagonist.

Features and Benefits

This compound was developed by Celgene. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

Packaging

1 g in glass bottle

100, 250 mg in glass bottle

25 mg in poly bottle

antibiotic activity spectrumfungi
formpowder
Gene Informationhuman ... GRIN1(2902), GRIN2A(2903), GRIN2B(2904), GRIN2C(2905), GRIN2D(2906), GRINA(2907), NOS1(4842), NOS2(4843), NOS2B(201288), NOS2C(645740), NOS3(4846)
InChI keyYBVNFKZSMZGRAD-UHFFFAOYSA-N
InChI1S/C19H24N4O2.2C2H6O4S/c20-18(21)14-4-8-16(9-5-14)24-12-2-1-3-13-25-17-10-6-15(7-11-17)19(22)23;2*3-1-2-7(4,5)6/h4-11H,1-3,12-13H2,(H3,20,21)(H3,22,23);2*3H,1-2H2,(H,4,5,6)
mode of actionenzyme | inhibits
mp188-194 °C (lit.)
originatorCelgene
Quality Level100
SMILES stringOCCS(O)(=O)=O.OCCS(O)(=O)=O.NC(=N)c1ccc(OCCCCCOc2ccc(cc2)C(N)=N)cc1
storage temp.−20°C
Cas Number140-64-7
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