Gallamine triethiodide, >=98% (TLC), powder, muscarinic receptor antagonist

Code: G8134-5G D2-231

Application

Gallamine triethiodide has been used:as a relaxant for measuring spinal trigeminal nucleus recordings from single neurons.as an antagonist in neuroblastoma cells ...


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€170.81 5G
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Application

Gallamine triethiodide has been used:as a relaxant for measuring spinal trigeminal nucleus recordings from single neurons.as an antagonist in neuroblastoma cells as M2 receptorto reduce eye movement during retinal surgery in rat

Biochem/physiol Actions

Gallamine triethiodide has anti-muscarinic effect. It is a competitive antagonist for the muscarinic receptor. Gallamine is regarded as neuromuscular blocking agent.

Muscle relaxant; allosteric muscarinic receptor antagonist with an order of potency of M2 > M1 = M4 > M3 = M5. Ligand for the peripheral anionic binding site of acetylcholinesterase.

Caution

Hygroscopic

Features and Benefits

This compound is featured on the Acetylcholine Receptors (Muscarinic) page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

This compound is a featured product for Neuroscience research. Click here to discover more featured Neuroscience products. Learn more about bioactive small molecules for other areas of research at sigma.com/discover-bsm.

Packaging

5, 25 g in poly bottle

assay≥98% (TLC)
formpowder
Gene Informationhuman ... CHRM1(1128), CHRM2(1129), CHRM3(1131), CHRM4(1132), CHRM5(1133), CHRNA1(1134), CHRNB1(1140), CHRND(1144), CHRNE(1145), CHRNG(1146)
InChI keyREEUVFCVXKWOFE-UHFFFAOYSA-K
InChI1S/C30H60N3O3.3HI/c1-10-31(11-2,12-3)22-25-34-28-20-19-21-29(35-26-23-32(13-4,14-5)15-6)30(28)36-27-24-33(16-7,17-8)18-9;;;/h19-21H,10-18,22-27H2,1-9H3;3*1H/q+3;;;/p-3
mp235 °C (dec.) (lit.)
Quality Level200
SMILES string[I-].[I-].[I-].CC[N+](CC)(CC)CCOc1cccc(OCC[N+](CC)(CC)CC)c1OCC[N+](CC)(CC)CC
solubilityethanol: soluble, H2O: 100 mg/mL
storage temp.2-8°C
Cas Number65-29-2
This product has met the following criteria to qualify for the following awards:



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