D-Val-Phe-Lys Chloromethyl Ketone; Dihydrochloride

Biochem/physiol Actions

Cell permeable: no

Reversible: no

Product does not compete with ATP.

Primary TargetHuman plasmin

Target IC₅₀: 100 pM for human plasmin

General description

Selective irreversible inhibitor of plasmin with high selectivity for plasmin over urokinase.

Selective irreversible inhibitor of plasmin with high selectivity for plasmin (IC₅₀ = 100 pM for human plasmin) over urokinase.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Other Notes

Woessner, J.F., Jr., et al. 1989. Steroids54, 491.

Packaging

Packaged under inert gas

5 mg in Plastic ampoule

Reconstitution

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.r>r>r>r>From Catalog:r>Desc. Field- added "(IC₅₀ = 100 pM for human plasmin) "

Sequence

H-D-Val-Phe-Lys-CMK

Warning

Toxicity: Standard Handling (A)