Biochem/physiol Actions
Target Ki: 130 nM against human MMP-3
Reversible: no
Primary Targethuman MMP-3
Product does not compete with ATP.
Cell permeable: yes
General description
A potent and cell-permeable inhibitor of human MMP-3 (Ki = 130 nM).
A cell-permeable, potent inhibitor of human MMP-3 (stromelysin; Ki = 130 nM).
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Other Notes
Kato, N., et al. 2002. Genome Informatics13, 272.MacPherson, L.J., et al. 1997. J. Med. Chem. 40, 2525.
Packaging
5 mg in Plastic ampoule
Reconstitution
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Warning
Toxicity: Standard Handling (A)
This product has met the following criteria to qualify for the following awards: