U-69593, solid

Code: U103-5MG D2-231

Biochem/physiol Actions

U-69593 is a selective κ opioid receptor agonist. U-69593 is known to inhibit cocaine sensitization in meso-limbic dopamine neurons by normalizing bas...


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€248.50 5MG
€305.66 inc. VAT
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Biochem/physiol Actions

U-69593 is a selective κ opioid receptor agonist. U-69593 is known to inhibit cocaine sensitization in meso-limbic dopamine neurons by normalizing basal overflow of dopamine.

Features and Benefits

This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Packaging

5 mg in glass bottle

25 mg in poly bottle

Preparation Note

U-69593 is soluble in 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin (10 mg/ml), 0.1 M HCl (>40 mg/ml), and ethanol (>40 mg/ml). However, it is insoluble in 0.1 M NaOH and water.

colorwhite
formsolid
Gene Informationhuman ... OPRD1(4985), OPRK1(4986), OPRM1(4988)mouse ... Oprk1(18387)rat ... Oprd1(24613), Oprk1(29335), Oprm1(25601)
InChI keyPGZRDDYTKFZSFR-ONTIZHBOSA-N
InChI1S/C22H32N2O2/c1-23(21(25)16-18-8-3-2-4-9-18)19-10-12-22(11-7-15-26-22)17-20(19)24-13-5-6-14-24/h2-4,8-9,19-20H,5-7,10-17H2,1H3/t19-,20-,22-/m0/s1
optical activity[α]/D +7.8°, c = 0.825 in methanol(lit.)
Quality Level100
SMILES stringCN([C@H]1CC[C@@]2(CCCO2)C[C@@H]1N3CCCC3)C(=O)Cc4ccccc4
solubility0.1 M NaOH: insoluble, 0.1 M HCl: >40 mg/mL, ethanol: >40 mg/mL, 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 10 mg/mL, H2O: insoluble
storage temp.2-8°C
Cas Number96744-75-1
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