PKS21004

Code: SML2445-5MG D2-231

Biochem/physiol Actions

PKS21004 is highly selective, potent and reversible inhibitor of the Plasmodium falciparum proteasome (Pf20S) β5 subunit. It is not active agains...


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€74.20 5MG
€91.27 inc. VAT
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Biochem/physiol Actions

PKS21004 is highly selective, potent and reversible inhibitor of the Plasmodium falciparum proteasome (Pf20S) β5 subunit. It is not active against mammalian c-20S and i-20S proteasome subunits. PKS21004 is effective against erythrocytic, sexual, and liver-stage parasites. Also it is active against parasites resistant to current antimalarials, and strains from patients in Africa.

assay≥98% (HPLC)
colorwhite to beige
formpowder
SMILES stringO=C(N[C@@H](CC(NC(C)(C)C)=O)C(NCCNC(C1=CC=CC(C2=CC=CC=C2)=C1)=O)=O)CCC3=CC=CC=C3
solubilityDMSO: 2 mg/mL, clear
storage temp.2-8°C
Cas Number2095521-90-5
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