MS417

Code: SML2442-5MG D2-231

Biochem/physiol Actions

MS417, a (+)-JQ1 analog, is a potent inhibitor of bromodomain-containing protein 4 (BRD4) that is highly specific for BRD4-BD1 and BRD4-BD2. MS417 bin...


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€137.70 5MG
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Biochem/physiol Actions

MS417, a (+)-JQ1 analog, is a potent inhibitor of bromodomain-containing protein 4 (BRD4) that is highly specific for BRD4-BD1 and BRD4-BD2. MS417 binds with similar affinity to BRD4-BD1 and BRD4-BD2 (Kd =36.1, and 25.4 nM), while bulky tBu of JQ1 prevents tight binding to the cavity at BD1.

assay≥98% (HPLC)
colorwhite to very dark brown
formpowder
SMILES stringO=C(OC)C[C@H]1C2=NN=C(C)N2C3=C(C(C)=C(C)S3)C(C4=CC=C(Cl)C=C4)=N1
solubilityDMSO: 2 mg/mL, clear
storage temp.2-8°C
Cas Number916489-36-6
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