CMPPE

Code: SML1584-25MG D2-231

Biochem/physiol Actions

CMPPE is a GABAB receptor positive allosteric modulator (PAM). GABAB receptor positive allosteric modulators have potential for treatment of many neur...


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€302.28 25MG
€371.80 inc. VAT
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Biochem/physiol Actions

CMPPE is a GABAB receptor positive allosteric modulator (PAM). GABAB receptor positive allosteric modulators have potential for treatment of many neuro-psychiatric disorders as well as drug dependence and seizures. The receptor is a GPCR expressed throughout the CNS; it acts as both an auto-receptor and heteroreceptor to mudulate GABA release and regulate K+ channels and Ca++ channels. CMPPE has the highest hypoactivity/anticonvulsant ratio.

Packaging

5, 25 mg in glass bottle

assay≥95% (HPLC)
colorwhite to light brown
formpowder
InChI keyTZWSGOPCLUTFBZ-UHFFFAOYSA-N
InChI1S/C20H23ClN4O/c1-14-12-20(24-10-3-2-4-17(24)9-11-26)25-19(22-14)13-18(23-25)15-5-7-16(21)8-6-15/h5-8,12-13,17,26H,2-4,9-11H2,1H3
Quality Level100
SMILES stringClC(C=C1)=CC=C1C2=NN(C(N3C(CCO)CCCC3)=CC(C)=N4)C4=C2
solubilityDMSO: 5 mg/mL, clear (warmed)
storage temp.2-8°C
Cas Number841253-81-4
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