MLS1547

Code: SML1331-5MG D2-231

Biochem/physiol Actions

MLS1547 is a highly efficacious D2 dopamine receptor (D2R) G protein-biased agonist that does not recruit β-arrestin, and is an antagonist of dop...


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€128.40 5MG
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Biochem/physiol Actions

MLS1547 is a highly efficacious D2 dopamine receptor (D2R) G protein-biased agonist that does not recruit β-arrestin, and is an antagonist of dopamine-stimulated β-arrestin recruitment to the D2 receptor. MLS-1547 is the first D2 receptor agonist with close to full efficacy for G protein signaling (EC50 = 370 nM), but no ability to recruit β-arrestin.

Packaging

5, 25 mg in glass bottle

assay≥98% (HPLC)
colorwhite to beige
formpowder
InChI keyOPEJNANYABTIGC-UHFFFAOYSA-N
InChI1S/C19H19ClN4O/c20-16-12-14(19(25)18-15(16)4-3-7-22-18)13-23-8-10-24(11-9-23)17-5-1-2-6-21-17/h1-7,12,25H,8-11,13H2
Quality Level100
SMILES stringOC1=C(CN2CCN(C3=NC=CC=C3)CC2)C=C(Cl)C4=CC=CN=C41
solubilityDMSO: 5 mg/mL, clear (warmed)
storage temp.2-8°C
Cas Number315698-36-3
Hazard Class6.1
Un Number2811
Pack GroupIII
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