Biochem/physiol Actions
Reversible: yes
Primary TargetD4
General description
A selective D4 dopamine receptor agonist (Ki = 8.7 nM, EC50 = 8.3 nM). Suitable for central and peripheral delivery. Used in studies of penile erection, learning and memory. Exibits some binding affinity towards human D2 and D3 Receptors (Ki = 2.8 µM).
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Other Notes
Melis, M. R. et al. 2005. Neurosci. Lett.379, 59.Bernaerts, P. et al. 2003. Behav. Brain Res.142, 41.
Packaging
10 mg in Glass bottle
Reconstitution
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Warning
Toxicity: Standard Handling (A)
This product has met the following criteria to qualify for the following awards: