05-23-3831-5MG Display Image

BQ-123, SODIUM SALT 1PC X 5MG

Code: 05-23-3831-5MG D2-231

Biochem/physiol Actions

Cell permeable: no

Reversible: no

Product does not compete with ATP.

Primary TargetETA (endothelin) receptor antagonist

Target...


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Your Price
€702.00 EACH
Discontinued

Biochem/physiol Actions

Cell permeable: no

Reversible: no

Product does not compete with ATP.

Primary TargetETA (endothelin) receptor antagonist

Target Ki: 40 nM for ETA versus 2.5 µM for ETB

General description

A highly potent, selective, and competitive ETA (endothelin) receptor antagonist (Ki = 40 nM for ETA versus Ki = 2.5 µM for ETB).

A highly potent and selective ETA (endothelin) receptor antagonist (Ki = 40 nM for ETA versus 2.5 µM for ETB).

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Other Notes

Nambi, P., et al. 1996. J. Pharmacol. Exp. Ther.277, 1567.Bax, W.A., and Saxena, P.R. 1994. Trends Pharmacol. Sci. 15, 379.Ihara, M., et al. 1991. Biochem. Biophys. Res. Commun. 178, 132.

Packaging

Yes

Physical form

Supplied as a sodium salt. Sold on the basis of peptide content.

Sequence

Cyclo(D-Asp-Pro-D-Val-Leu-D-Trp, Na)

Warning

Toxicity: Standard Handling (A)

assay≥95% (HPLC)
colorwhite
formsolid
manufacturer/tradenameCalbiochem®
Quality Level100
shipped inambient
solubilitywater: 1 mg/mL
storage conditiondesiccated (hygroscopic), OK to freeze
storage temp.−20°C
Code
Description
Unit Size
List Price
Qty
05-23-3831-1MG
Unit:EACH
List Price: €221.54
Source:List Price
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