FOSAPREPITANT DIMEGLUMINE

Code: SML2228-10MG D2-231

Biochem/physiol Actions

Fosaprepitant dimeglumine is a Substance P/neurokinin-1 (NK1) receptor antagonist. It is a water soluble prodrug of the antiemetic drug aprepitant.

read more

Your Price
€93.20 10MG
€114.64 inc. VAT
REQUEST

Biochem/physiol Actions

Fosaprepitant dimeglumine is a Substance P/neurokinin-1 (NK1) receptor antagonist. It is a water soluble prodrug of the antiemetic drug aprepitant.

Fosaprepitant dimeglumine acts as a therapeutic agent to treat chemotherapy-induced nausea and vomiting. It also acts as a weak inhibitor of cytochrome P450 3A4 (CYP3A4).

assay≥98% (HPLC)
colorwhite to beige
formpowder
optical activity[α]/D +27 to +34°, c = 0.5 in methanol
shipped inwet ice
SMILES stringFC1=CC=C([C@@H]2N(CCO[C@@H]2O[C@@H](C3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3)C)CC(NC4=O)=NN4P(O)(O)=O)C=C1.CNC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O
solubilityH2O: 2 mg/mL, clear
storage conditiondesiccated
storage temp.−20°C
This product has met the following criteria to qualify for the following awards:



PROCEED TO CHECKOUT

HAVE AN ACCOUNT? LOGIN

GUEST CHECKOUT

Proceed as a guest. You will have the option to register to access exclusive pricing and stock availability features after checkout.