VPC-13566

Code: SML1886-5MG D2-231

Biochem/physiol Actions

VPC-13566 is Binding Function 3 (BF3)-specific inhibitor of the androgen receptor. VPC-13566 potently inhibits AR transcriptional activity by displace...


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€127.40 5MG
€156.70 inc. VAT
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Biochem/physiol Actions

VPC-13566 is Binding Function 3 (BF3)-specific inhibitor of the androgen receptor. VPC-13566 potently inhibits AR transcriptional activity by displacement of the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines including an enzalutamide-resistant cell line and inhibits the growth of AR-dependent prostate cancer xenograft in mice.

Packaging

5, 25 mg in glass bottle

assay≥98% (HPLC)
colorwhite to beige
formpowder
Quality Level100
SMILES stringCC1=CC=CC2=C1NC=C2C3=NC4=CC=CC=C4C=C3
solubilityDMSO: 20 mg/mL, clear
storage temp.2-8°C
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