Biochem/physiol Actions

Cell permeable: no

Reversible: no

Product does not compete with ATP.

Primary Targeturokinase

Target IC₅₀: ﹤1 µM against urokinase

General description

An irreversible inhibitor of urokinase (IC₅₀﹤1 µM) and Factor Xa.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Other Notes

Kettner, C., and Shaw, E. 1979. Biochim. Biophys. Acta569, 31.

Packaging

5 mg in Plastic ampoule

Reconstitution

Following reconstitution aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C. Avoid freeze/thaw cycles of stock solution.

Sequence

H-Glu-Gly-Arg-CMK

Warning

Toxicity: Standard Handling (A)