CTOP

Code: 5080150001 D2-231

Biochem/physiol Actions

Primary Targetmu opioid

General description

A potent antagonist highly selective for µ opioid receptor (Ki

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€190.50 EACH
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Biochem/physiol Actions

Primary Targetmu opioid

General description

A potent antagonist highly selective for µ opioid receptor (Ki = 0.96 nM for µ receptor and >10,000 nM for δ receptors). Often used for studying the functional roles of µ opioid receptors in both central and peripheral nervous systems.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Other Notes

Feng, Y., et al. 2012. Curr Drug Targets.13, 230.Hawkins, N., et al. 1989. J. Pharmacol. Exp. Ther.248, 73.Gulya, K., et al. 1988. Eur. J. Pharmacol.150, 355.

Packaging

1 mg in Glass bottle

Physical form

Supplied as trifluoracetate salt

Sequence

D-Phe-Cys-Tyr-D-Trp-Orn-Thr-Pen-Thr-NH2 (Orn: ornithine; Pen: penicillamine; SS bond: 2-7)

Warning

Toxicity: Standard Handling (A)

assay≥98% (HPLC)
colorwhite
formsolid
InChI keyPZWWYAHWHHNCHO-UHFFFAOYSA-N
InChI1S/C50H67N11O11S2/c1-26(62)39(42(53)65)59-49(72)41-50(3,4)74-73-25-38(58-43(66)33(52)21-28-11-6-5-7-12-28)47(70)56-36(22-29-16-18-31(64)19-17-29)45(68)57-37(23-30-24-54-34-14-9-8-13-32(30)34)46(69)55-35(15-10-20-51)44(67)60-40(27(2)63)48(71)61-41/h5-9,11-14,16-19,24,26-27,33,35-41,54,62-64H,10,15,20-23,25,51-52H2,1-4H3,(H2,53,65)(H,55,69)(H,56,70)(H,57,68)(H,58,66)(H,59,72)(H,60,67)(H,61,71)
manufacturer/tradenameCalbiochem®
potency0.96 nM Ki
Quality Level100
solubilitywater: soluble
storage conditionprotect from light, OK to freeze
storage temp.−20°C
Cas Number103429-31-8
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